Hexarelinumest syntheticumpeptidum secretagogum hormonis crescentis (GHS)et potensAgonista GHSR-1a, elaboratum ad stimulandumemissio hormonis crescentis endogeni (GH)Ad id pertinetfamilia mimetica ghrelinorumet ex sex aminoacidis (hexapeptido) constat, stabilitatem metabolicam auctam et effectus GH-liberantes fortiores praebens, comparatione facta cum analogis prioribus sicut GHRP-6.
Hexarelinum late investigatur propter usus suos inendocrinologia, atrophia musculorum, reparatio cardiaca, et therapiae contra senectutem, propter facultatem suam naturaliter GH elevandi etfactor crescendi insulinum similis 1 (IGF-1)gradus sine directe introductione hormonum externorum.
Hexarelinum se adhaeretreceptor secretagogi hormonis crescentis (GHSR-1a)in pituitaria et hypothalamo, actionem imitansghrelinum—fames naturalis corporis et hormon GH liberans.
Actiones physiologicae principales:
Emissionem GH pulsatilem stimulat
Augmentat circulationemIGF-1gradus
Promoveteffectus anabolici(incrementum musculorum, recuperatio)
Sustentatmetabolismus adipumetregeneratio cellularum
Exhibeatur fortassecardioprotegensetanti-apoptoticuseffectus
Dissimilis quibusdam aliis peptidis GHS, Hexarelin facit...non significanter auget cortisol aut prolactin, profilum endocrini mundiorem offerens.
Promovetmassa corporis macraprogressus
Augmentatreparatio et regeneratio musculorum
Studium insarcopenia, cachexiaet recuperatio post chirurgicam
Studia praeclinica ostenduntfunctio cardiaca emendatapost laesionem myocardii
Reducitfibrosis cardiacaet augetfractio ejectionis ventriculi sinistri
Usus potentialis ininsufficientia cordisetsenescentia cardiacaexempla
Incrementumlipolysiset emendatsensibilitas insulini
Sustentatcurationes contra senectutemper stimulationem axis GH/IGF-1
Fortasse adiuvabit conservaredensitas ossium et salus articulationum
Puritas ≥ 99%
Productum persynthesis peptidorum in phase solida (SPPS)
Normae similes GMP, endotoxini et residua solventium humilia
Copia flexibilis:Investigatio et progressio ad scalam commercialem